Search results for "hirshfeld surface"

showing 10 items of 41 documents

Crystal structure, Hirshfeld analysis and molecular docking with the vascular endothelial growth factor receptor-2 of (3Z)-5-fluoro-3-(hydroxyimino)i…

2017

The reaction between 5-fluoroisatin and hydroxylamine hydrochloride in acidic ethanol yields the title compound, C8H5FN2O2, whose molecular structure matches the asymmetric unit and is nearly planar with an r.m.s. deviation for the mean plane through all non-H atoms of 0.0363 Å. In the crystal, the molecules are linked by N—H...N, N—H...O and O—H...O hydrogen-bonding interactions into a two-dimensional network along the (100) plane, forming rings withR22(8) andR12(5) graph-set motifs. The crystal packing also features weak π–π interactions along the [100] direction [centroid-to-centroid distance 3.9860 (5) Å]. Additionally, the Hirshfeld surface analysis indicates that the major contributio…

0301 basic medicinecrystal structureChemistryStereochemistryGeneral ChemistryIndolin 2 oneCrystal structure010403 inorganic & nuclear chemistryCondensed Matter Physics01 natural sciences0104 chemical scienceslcsh:Chemistry03 medical and health sciencesCrystallography030104 developmental biologyisatin derivative–VEGFR-2 in silico evaluationlcsh:QD1-999Docking (molecular)MoleHirshfeld surface analysisGeneral Materials ScienceActa Crystallographica Section E Crystallographic Communications
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Crystal structure of (3E)-5-nitro-3-(2-phenylhydrazinylidene)-1H-indol-2(3H)-one

2017

The reaction between 5-nitroisatin and phenylhydrazine in acidic ethanol yields the title compound, C14H10N4O3, whose molecular structure deviates slightly from a planar geometry (r.m.s. deviation = 0.065 Å for the mean plane through all non-H atoms). An intramolecular N—H...O hydrogen bond is present, forming a ring of graph-set motifS(6). In the crystal, molecules are linked by N—H...O and C—H...O hydrogen-bonding interactions into a two-dimensional network along (120), and rings of graph-set motifR22(8),R22(26) andR44(32) are observed. Additionally, a Hirshfeld surface analysis suggests that the molecules are stacked along [100] through C=O...Cginteractions and indicates that the most im…

0301 basic medicinecrystal structureStereochemistryin silico evaluationtwo-dimensional hydrogen-bonded networkCrystal structureReductaseisatin–hydrazone derivative010403 inorganic & nuclear chemistryRing (chemistry)01 natural sciencesCrystal03 medical and health scienceschemistry.chemical_compoundHirshfeld surface calculationGeneral Materials ScienceCrystallographybiologyHydrogen bondActive siteGeneral ChemistryCondensed Matter Physics0104 chemical sciences030104 developmental biologychemistryQD901-999biology.proteinNitroisatin-hydrazone derivativeDerivative (chemistry)Acta Crystallographica Section E: Crystallographic Communications
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The effect of the fused-ring substituent on anthracene chalcones: crystal structural and DFT studies of 1-(anthracen-9-yl)-3-(naphthalen-2-yl)prop-2-…

2018

Two new anthracene chalcones, namely 1-(anthracen-9-yl)-3-(naphthalen-2-yl)prop-2-en-1-one and 1-(anthracen-9-yl)-3-(pyren-1-yl)prop-2-en-1-one, have been successfully synthesized and the effect of the different fused ring substituent system attached to the anthracene chalcone derivative investigated. These compounds show a very narrow band gap due to the large p-conjugated systems, making them promising candidates as optoelectronic materials. Hirshfeld surface analysis has been carried out to show the contribution of inter­molecular contacts and weak inter­actions to supra­molecular stabilization.

Chalconecrystal structureSubstituentchalconeCrystal structure010402 general chemistry010403 inorganic & nuclear chemistryRing (chemistry)01 natural sciencesMedicinal chemistryDFTResearch Communicationschemistry.chemical_compoundMoietyGeneral Materials ScienceAnthraceneCrystallographyHirshfeld surfaceUV-VisGeneral ChemistryCondensed Matter Physics0104 chemical scienceschemistryQD901-999Density functional theoryEnoneActa crystallographica. Section E, Crystallographic communications
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Primary- and secondary-octahedral distortion factors in bis(1,4-H2-1,2,4-triazolium) pentabromidoantimonate(III) –1,4-H2-1,2,4-triazolium bromide

2015

Abstract The analysis of octahedral distortion in the structure of inorganic–organic (C2H4N3)2[SbBr5]·(C2H4N3)Br (BTPTB) bromidoantimonate(III) determined at 295 and 85 K, supported by the Hirshfeld surface analysis and the data retrieved from the Cambridge Structural Database, is presented. The anionic substructure of BTPTB is built from distorted [SbBr6]3− octahedra that are connected by the cis corners forming polymeric one-dimensional [{SbBr5}n]2n− zig-zag chains running parallel to the a axis and isolated Br− ions. The organic substructure consists of the fully ordered 1,4-H2-1,2,4-triazolium cations. The oppositely charged substructures are linked by the system of N(C)–H⋯Br hydrogen b…

ChemistryHydrogen bondIonHybrid materials; Octahedral distortion; Hirshfeld surface analysis; Distortion parameters; Hydrogen bondingInorganic Chemistrychemistry.chemical_compoundCrystallographyOctahedronBromideDistortionOctahedral molecular geometryMaterials ChemistrySubstructurePhysical and Theoretical ChemistryHybrid materialPolyhedron
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Crystal structure and Hirshfeld surface analysis of (E)-4-chloro-N-{2-[2-(4-nitro­benzyl­idene)hydrazin-1-yl]-2-oxoeth­yl}benzene­sulfonamide N,N-di­…

2018

Reaction of N-(4-chloro­benzene­sulfon­yl)glycinyl hydrazide with 4-nitro­benzaldehyde gives the N,N-di­methyl­formamide monosolvated N-acyl­hydrazone derivative, (E)-N-{2-[2-(4-nitro­benzyl­idene)- hydrazine-1-yl]-2-oxoeth­yl}-4-χhloro­benzene­sulfonamide. Rings of (10) and (11) graph-set motifs are formed in the crystal structure by N—H⋯O and C—H⋯O hydrogen bonds. The two-dimensional fingerprint (FP) plots for significant inter­molecular inter­actions indicate that the greatest contribution is from the O⋯H/H⋯O contacts (31.3%), corresponding to N⋯H⋯O/C⋯H⋯O inter­actions.

Formamidecrystal structureHydrazoneCrystal structureDihedral angle010402 general chemistry010403 inorganic & nuclear chemistryRing (chemistry)01 natural sciencesMedicinal chemistryResearch Communicationslcsh:Chemistrychemistry.chemical_compoundhydrazoneHirshfeld surface analysisGeneral Materials Sciencechemistry.chemical_classificationSchiff baseHydrogen bondinter­molecular hydrogen bondsAromaticityGeneral ChemistryCondensed Matter Physics0104 chemical sciencesintermolecular hydrogen bondslcsh:QD1-999chemistryinversion dimersActa Crystallographica Section E: Crystallographic Communications
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X-ray Single Crystal Structure, Tautomerism Aspect, DFT, NBO, and Hirshfeld Surface Analysis of a New Schiff Bases Based on 4-Amino-5-Indol-2-yl-1,2,…

2021

Four different new Schiff basses tethered indolyl-triazole-3-thione hybrid were designed and synthesized. X-ray single crystal structure, tautomerism, DFT, NBO and Hirshfeld analysis were explored. X-ray crystallographic investigations with the aid of Hirshfeld calculations were used to analyze the molecular packing of the studied systems. The H···H, H···C, S···H, Br···C, O···H, C···C and N···H interactions are the most important in the molecular packing of 3. In case of 4, the S···H, N···H, S···C and C···C contacts are the most significant. The results obtained from the DFT calculations indicated that the thione tautomer is energetically lower than the thiol one by 13.9545 and 13.7464 kcal…

General Chemical Engineeringtautomerism aspectInorganic Chemistrysymbols.namesakeGeneral Materials SciencetyppiyhdisteetDebyechemistry.chemical_classificationkemiallinen synteesiCrystallographyX-rayCondensed Matter Physicsindolyl-triazole-3-thioneTautomerSchiff bases; indolyl-triazole-3-thione; tautomerism aspect; Hirshfeld Surface AnalysisCrystallographyDipolechemistryQD901-999Thiolsymbols1 2 4 triazole 3 thioneSchiff basesHirshfeld Surface AnalysisSingle crystaltautomeriaNatural bond orbitalCrystals; Volume 11; Issue 9; Pages: 1041
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Synthesis and X-ray Crystal Structure Analysis of Substituted 1,2,4-Triazolo [4’,3’:2,3]pyridazino[4,5-b]indole and Its Precursor

2023

The hit compound 1,2,4-triazolo[4’,3’:2,3]pyridazino[4,5-b]indole 3 was synthesized from the reflux of 4-amino-5-indolyl-1,2,4-triazole-3-thione 1 with 4′-bromoacetophenone 2 in methanol catalyzed by concentrated HCl and the desired final molecule was obtained by recrystallization from methanol. The suggested structures of compounds 1 and 3 based on the spectral characterizations were confirmed by X-ray single crystal diffraction analysis. Compound 3 crystallized in the triclinic crystal system and P-1 space group with a = 5.9308(2) Å, b = 10.9695(3) Å, c = 14.7966(4) Å, α = 100.5010(10)°, β = 98.6180(10)°, and γ = 103.8180(10)°. On the other hand, the crystal system of 1 is monoclinic, whe…

Hirshfeld surface analysispyridazinesindoleskidetiedekiteetpintakemiaröntgenkristallografiapyridazino[45-b]indol-4-oneX-ray single crystal
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Temperature-dependent polymorphism of N-(4-fluorophenyl)-1,5-dimethyl-1H-imidazole-4-carboxamide 3-oxide: experimental and theoretical studies on int…

2014

X-ray analysis of N-(4-fluorophenyl)-1,5-dimethyl-1H-imidazole-4-carboxamide 3-oxide reveals the temperature-dependent polymorphism associated with the crystallographic symmetry conversion. The observed crystal structure transformation corresponds to a symmetry reduction from I41 /a (I) to P43 (II) space groups. The phase transition mainly concerns the subtle but clearly noticeable reorganization of molecules in the crystal space, with the structure of individual molecules left almost unchanged. The Hirshfeld surface analysis shows that various intermolecular contacts play an important role in the crystal packing, revealing graphically the differences in spatial arrangements of the molecule…

Hydrogen bondingCrystallographic point groupAIM approachHydrogen bondChemistryIntermolecular forceCrystal structureCondensed Matter PhysicsAcceptorN-oxideX-ray diffractionCrystallographyPolymorphism (materials science)Intramolecular forceMoleculeHirshfeld surface analysisPhysical and Theoretical ChemistryPolymorphism
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Synthesis, X-ray Structure of Two Hexa-Coordinated Ni(II) Complexes with s-Triazine Hydrazine Schiff Base Ligand

2023

The hydrazine s-triazine ligand (E)-4,4’-(6-(2-(1-(pyridin-2-yl)ethylidene)hydrazinyl)-1,3,5-triazine-2,4-diyl)dimorpholine (DMPT) was used to synthesize two new Ni(II) complexes via a self-assembly technique. The two complexes were synthesized by a one-pot synthesis strategy and characterized by elemental analysis, FTIR and single-crystal X-ray diffraction analysis to be [Ni(DMPT)(H2O)3](NO3)2.3H2O (1) and [Ni(DMPT)(H2O)3](NO3)2.H2O (2). The structures of both complexes were very similar regarding the coordination sphere and counter anions, but differ only in the number of the crystal water molecules. In the case of complex 1, there are three water molecules instead of one H2O molecu…

Inorganic ChemistryX-rayantimikrobiset yhdisteetNi(II) complexesmolecular packings-triazine hydrazoneHirshfeld surfaceantimicrobialkompleksiyhdisteetnikkeli<i>s</i>-triazine hydrazone; molecular packing; X-ray; Ni(II) complexes; Hirshfeld surface; antimicrobialröntgenkristallografia
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Isostructural Inorganic–Organic Piperazine-1,4-diium Chlorido- and Bromidoantimonate(III) Monohydrates: Octahedral Distortions and Hydrogen Bonds

2020

Halogenidoantimonate(III) monohydrates of the (C4H12N2)[SbX5]&middot

Models Molecularcrystal structureMaterials scienceHydrogenSurface PropertiesMolecular ConformationPharmaceutical Sciencechemistry.chemical_elementCrystal structurelow temperatureArticleAnalytical Chemistrylcsh:QD241-441lcsh:Organic chemistryDrug DiscoveryMoleculeHirshfeld surface analysisPhysical and Theoretical ChemistryIsostructuralOrganic Chemicalsoctahedral distortionPiperazineHydrogen bondOrganic Chemistryhydrogen bondinginorganic–organic hybrid materialsCrystallographyOctahedronchemistryChemistry (miscellaneous)Inorganic ChemicalsMolecular MedicineWater of crystallizationhalogenidoantimonates(III)Monoclinic crystal systemMolecules
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